Product name: Chelerythrine
Plant source: Toddalia asiatica (L.)Lam.
Molecular formula: C21H18ClNO4
Molecular weight: 383.83
Construction:
CAS: 34316-15-9 .
Characteristics: light yellow powder or white powder, melting point:
195-205°C , 207℃(lmol ethanol) or 250℃(0.5mol water)
Specifications: 50％、90%、95%、98％ HPLC
Biological Activity:
Potent, cell-permeable inhibitor of protein kinase C (IC50 = 660 nM);
competitive with respect to the phosphate acceptor and non-competitive
with respect to ATP. Has a wide range of biological activities,
including antiplatelet, anti-inflammatory, antibacterial and antitumor
effects. Activates MAPK pathways, independent of PKC inhibition.
Inhibits binding of BclXL to Bak (IC50 = 1.5 μM) or Bad proteins and
stimulates apoptosis.
Packing: 1kg/ aluminum bag
25kgs/ fiber durm or according to customer's demand
Shelf life: 2 years
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